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PDB Identifier Description Ligand Receptor SCOP pdb.org
3GYT Nuclear receptor DAF-12 from parasitic nematode Strongyloides stercoralis in complex with its physiological ligand dafachronic acid delta 4 B A
3H0A Crystal Structure of Peroxisome Proliferator-Activated Receptor Gamma (PPARg) and Retinoic Acid Receptor Alpha (RXRa) in Complex with 9-cis Retinoic Acid, Co-activator Peptide, and a Partial Agonist B A
3GYU Nuclear receptor DAF-12 from parasitic nematode Strongyloides stercoralis in complex with its physiological ligand dafachronic acid delta 7 B A
3G9E Aleglitaar. a new. potent, and balanced dual ppara/g agonist for the treatment of type II diabetes B A
3FXV Identification of an N-oxide pyridine GW4064 analogue as a potent FXR agonist B A
3G8I Aleglitazar, a new, potent, and balanced PPAR alpha/gamma agonist for the treatment of type II diabetes Z A
3FUR Crystal Structure of PPARg in complex with INT131 H A
3FUG Crystal Structure of the Retinoid X Receptor Ligand Binding Domain Bound to the Synthetic Agonist 3-[4-Hydroxy-3-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaphthalen-2-yl)-phenyl]acrylic Acid B A
3F9Z Structural Insights into Lysine Multiple Methylation by SET Domain Methyltransferases, SET8-Y245F / H4-Lys20 / AdoHcy G A
3F9W Structural Insights into Lysine Multiple Methylation by SET Domain Methyltransferases, SET8-Y334F / H4-Lys20 / AdoHcy F AB
3F7D SF-1 LBD bound by phosphatidylcholine B A
3ET3 Structure of PPARgamma with 3-[5-Methoxy-1-(4-methoxy-benzenesulfonyl)-1H-indol-3-yl]-propionic acid P A
3ET1 Structure of PPARalpha with 3-[5-Methoxy-1-(4-methoxy-benzenesulfonyl)-1H-indol-3-yl]-propionic acid P A
3EMW Crystal Structure of human splA/ryanodine receptor domain and SOCS box containing 2 (SPSB2) in complex with a 20-residue VASA peptide B A
3ECH The MarR-family repressor MexR in complex with its antirepressor ArmR C BA
3E94 Crystal structure of RXRalpha ligand binding domain in complex with tributyltin and a coactivator fragment B A
3E7C Glucocorticoid Receptor LBD bound to GSK866 D B
3DCG Crystal Structure of the HIV Vif BC-box in Complex with Human ElonginB and ElonginC F B POZ domain
3DAB Structure of the human Mdmx protein bound to the p53 tumor suppressor transactivation domain D C
3DAC Structure of the human Mdmx protein bound to the p53 tumor suppressor transactivation domain P M
3D9O Snapshots of the RNA processing factor SCAF8 bound to different phosphorylated forms of the Carboxy-Terminal Domain of RNA-Polymerase II Z B
3D8C Factor inhibiting HIF-1 alpha D201G mutant in complex with ZN(II), alpha-ketoglutarate and HIF-1 alpha 19mer B A
3D24 Crystal structure of ligand-binding domain of estrogen-related receptor alpha (ERRalpha) in complex with the peroxisome proliferators-activated receptor coactivator-1alpha box3 peptide (PGC-1alpha) B A Nuclear receptor ligand-binding domain
3D1F Crystal structure of E. coli sliding clamp (beta) bound to a polymerase III peptide P A DNA clamp
3D1E Crystal structure of E. coli sliding clamp (beta) bound to a polymerase II peptide P A DNA clamp
3CWD Molecular recognition of nitro-fatty acids by PPAR gamma C A Nuclear receptor ligand-binding domain
3CS8 Structural and Biochemical Basis for the Binding Selectivity of PPARg to PGC-1a B A Nuclear receptor ligand-binding domain
3CFS Structural basis of the interaction of RbAp46/RbAp48 with histone H4 E B
3C0T Structure of the Schizosaccharomyces pombe Mediator subcomplex Med8C/18 B A
3BQD Doubling the Size of the Glucocorticoid Receptor Ligand Binding Pocket by Deacylcortivazol B A Nuclear receptor ligand-binding domain
2ZXN A New Class of Vitamin D Receptor Ligands that Induce Structural Rearrangement of the Ligand-binding Pocket C A
3BEJ Structure of human FXR in complex with MFA-1 and co-activator peptide E A Nuclear receptor ligand-binding domain
2ZMJ Crystal Structure of Rat Vitamin D Receptor Bound to Adamantyl Vitamin D Analogs: Structural Basis for Vitamin D Receptor Antagonism and/or Partial Agonism C A Nuclear receptor ligand-binding domain
2ZMI Crystal Structure of Rat Vitamin D Receptor Bound to Adamantyl Vitamin D Analogs: Structural Basis for Vitamin D Receptor Antagonism and/or Partial Agonism C A Nuclear receptor ligand-binding domain
2ZMH Crystal Structure of Rat Vitamin D Receptor Bound to Adamantyl Vitamin D Analogs: Structural Basis for Vitamin D Receptor Antagonism and/or Partial Agonism C A Nuclear receptor ligand-binding domain
2ZL9 2-Substituted-16-ene-22-thia-1alpha,25-dihydroxy-26,27-dimethyl-19-norvitamin D3 analogs: Synthesis, biological evaluation and crystal structure C A Nuclear receptor ligand-binding domain
2ZLA 2-Substituted-16-ene-22-thia-1alpha,25-dihydroxy-26,27-dimethyl-19-norvitamin D3 analogs: Synthesis, biological evaluation and crystal structure C A Nuclear receptor ligand-binding domain
2ZLC 2-Substituted-16-ene-22-thia-1alpha,25-dihydroxy-26,27-dimethyl-19-norvitamin D3 analogs: Synthesis, biological evaluation and crystal structure C A Nuclear receptor ligand-binding domain
2ZFX Crystal structure of the rat vitamin D receptor ligand binding domain complexed with YR301 and a synthetic peptide containing the NR2 box of DRIP 205 C A
2Z34 Crystal structure of SpCia1/Asf1 complex with Hip1 C DA Immunoglobulin-like beta-sandwich
2Z32 Crystal structure of Keap1 complexed with Prothymosin alpha B A 6-bladed beta-propeller
2V52 STRUCTURE OF MAL-RPEL2 COMPLEXED TO G-ACTIN M A
2V51 STRUCTURE OF MAL-RPEL1 COMPLEXED TO ACTIN E A
2QZO Crystal Structure of the Estrogen Receptor Alpha Ligand Binding Domain Complexed with WAY-169916 C A
2QXV Structural basis of EZH2 recognition by EED B A
2QXM Crystal Structure of the Estrogen Receptor Alpha Ligand Binding Domain Complexed to Burned Meat Compound PhIP C A
2QSE Crystal Structure of the Estrogen Receptor Alpha Ligand Binding Domain complexed with Burned Meat Compound 4-OH-PhIP C A
2QR9 Crystal Structure of the Estrogen Receptor Alpha Ligand Binding Domain Complexed with an Oxabicyclic Derivative Compound C A
2QPY AR LBD with small molecule B A Nuclear receptor ligand-binding domain
2QGT Crystal Structure of the Estrogen Receptor Alpha Ligand Binding Domain Complexed to an Ether Estradiol Compound C A
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