Annotation 'Nuclear receptor ligand-binding domain'

Showing 1-50 of 75 results
PDB Identifier Description Ligand Receptor SCOP pdb.org
3ERD HUMAN ESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH DIETHYLSTILBESTROL AND A GLUCOCORTICOID RECEPTOR INTERACTING PROTEIN 1 NR BOX II PEPTIDE C A Nuclear receptor ligand-binding domain
3DCT FXR with SRC1 and GW4064 B A Nuclear receptor ligand-binding domain
3D24 Crystal structure of ligand-binding domain of estrogen-related receptor alpha (ERRalpha) in complex with the peroxisome proliferators-activated receptor coactivator-1alpha box3 peptide (PGC-1alpha) B A Nuclear receptor ligand-binding domain
3CWD Molecular recognition of nitro-fatty acids by PPAR gamma C A Nuclear receptor ligand-binding domain
3CS8 Structural and Biochemical Basis for the Binding Selectivity of PPARg to PGC-1a B A Nuclear receptor ligand-binding domain
3BQD Doubling the Size of the Glucocorticoid Receptor Ligand Binding Pocket by Deacylcortivazol B A Nuclear receptor ligand-binding domain
3BEJ Structure of human FXR in complex with MFA-1 and co-activator peptide E A Nuclear receptor ligand-binding domain
2ZMH Crystal Structure of Rat Vitamin D Receptor Bound to Adamantyl Vitamin D Analogs: Structural Basis for Vitamin D Receptor Antagonism and/or Partial Agonism C A Nuclear receptor ligand-binding domain
2ZMI Crystal Structure of Rat Vitamin D Receptor Bound to Adamantyl Vitamin D Analogs: Structural Basis for Vitamin D Receptor Antagonism and/or Partial Agonism C A Nuclear receptor ligand-binding domain
2ZMJ Crystal Structure of Rat Vitamin D Receptor Bound to Adamantyl Vitamin D Analogs: Structural Basis for Vitamin D Receptor Antagonism and/or Partial Agonism C A Nuclear receptor ligand-binding domain
2ZLC 2-Substituted-16-ene-22-thia-1alpha,25-dihydroxy-26,27-dimethyl-19-norvitamin D3 analogs: Synthesis, biological evaluation and crystal structure C A Nuclear receptor ligand-binding domain
2ZLA 2-Substituted-16-ene-22-thia-1alpha,25-dihydroxy-26,27-dimethyl-19-norvitamin D3 analogs: Synthesis, biological evaluation and crystal structure C A Nuclear receptor ligand-binding domain
2ZL9 2-Substituted-16-ene-22-thia-1alpha,25-dihydroxy-26,27-dimethyl-19-norvitamin D3 analogs: Synthesis, biological evaluation and crystal structure C A Nuclear receptor ligand-binding domain
2QPY AR LBD with small molecule B A Nuclear receptor ligand-binding domain
2Q7I The Wild Type Androgen Receptor Ligand Binding Domain Bound with Testosterone and an AR 20-30 Peptide B A Nuclear receptor ligand-binding domain
2Q7J The Wild Type Androgen Receptor Ligand Binding Domain Bound with Testosterone and a TIF2 box 3 Coactivator Peptide 740-753 B A Nuclear receptor ligand-binding domain
2P54 a crystal structure of PPAR alpha bound with SRC1 peptide and GW735 B A Nuclear receptor ligand-binding domain
2P1V Crystal structure of the ligand binding domain of the retinoid X receptor alpha in complex with 3-(2\'-propoxy)-tetrahydronaphtyl cinnamic acid and a fragment of the coactivator TIF-2 B A Nuclear receptor ligand-binding domain
2P1T Crystal structure of the ligand binding domain of the retinoid X receptor alpha in complex with 3-(2\'-methoxy)-tetrahydronaphtyl cinnamic acid and a fragment of the coactivator TIF-2 B A Nuclear receptor ligand-binding domain
2P1U Crystal structure of the ligand binding domain of the retinoid X receptor alpha in complex with 3-(2\'-ethoxy)-tetrahydronaphtyl cinnamic acid and a fragment of the coactivator TIF-2 B A Nuclear receptor ligand-binding domain
2OVH Progesterone Receptor with Bound Asoprisnil and a Peptide from the Co-Repressor SMRT B A Nuclear receptor ligand-binding domain
2O4R Crystal Structure of Rat Vitamin D Receptor Ligand Binding Domain Complexed with VitIII 17-20E and the NR2 Box of DRIP 205 C A Nuclear receptor ligand-binding domain
2O4J Crystal Structure of Rat Vitamin D Receptor Ligand Binding Domain Complexed with VitIII 17-20Z and the NR2 Box of DRIP 205 C A Nuclear receptor ligand-binding domain
2NV7 Crystal Structure of Estrogen Receptor Beta Complexed with WAY-555 C A Nuclear receptor ligand-binding domain
2J7Y STRUCTURE OF 17-EPIESTRIOL-BOUND ESTROGEN RECEPTOR BETA LBD IN COMPLEX WITH LXXLL MOTIF FROM NCOA5 B A Nuclear receptor ligand-binding domain
2J7X STRUCTURE OF ESTRADIOL-BOUND ESTROGEN RECEPTOR BETA LBD IN COMPLEX WITH LXXLL MOTIF FROM NCOA5 B A Nuclear receptor ligand-binding domain
2HFP Crystal Structure of PPAR Gamma with N-sulfonyl-2-indole carboxamide ligands B A Nuclear receptor ligand-binding domain
2GTK Structure-based Design of Indole Propionic Acids as Novel PPARag CO-Agonists B A Nuclear receptor ligand-binding domain
2GPO Estrogen Related Receptor-gamma ligand binding domain complexed with a synthetic peptide from RIP140 C A Nuclear receptor ligand-binding domain
2FVJ A novel anti-adipogenic partial agonist of peroxisome proliferator-activated receptor-gamma (PPARG) recruits pparg-coactivator-1 alpha (PGC1A) but potentiates insulin signaling in vitro B A Nuclear receptor ligand-binding domain
2AO6 Crystal structure of the human androgen receptor ligand binding domain bound with TIF2(iii) 740-753 peptide and R1881 B A Nuclear receptor ligand-binding domain
1ZGY Structural and Biochemical Basis for Selective Repression of the Orphan Nuclear Receptor LRH-1 by SHP B A Nuclear receptor ligand-binding domain
1YYE Crystal structure of estrogen receptor beta complexed with way-202196 C A Nuclear receptor ligand-binding domain
1XOW Crystal structure of the human androgen receptor ligand binding domain bound with an androgen receptor NH2-terminal peptide, AR20-30, and R1881 B A Nuclear receptor ligand-binding domain
1XB7 X-ray structure of ERRalpha LBD in complex with a PGC-1alpha peptide at 2.5A resolution P A Nuclear receptor ligand-binding domain
1X7J CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH GENISTEIN C A Nuclear receptor ligand-binding domain
1X7B CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH ERB-041 C A Nuclear receptor ligand-binding domain
1X78 CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH WAY-244 C A Nuclear receptor ligand-binding domain
1X76 CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH WAY-697 C A Nuclear receptor ligand-binding domain
1U9E CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH WAY-397 C A Nuclear receptor ligand-binding domain
1U3S Crystal Structure of Estrogen Receptor beta complexed with WAY-797 C A Nuclear receptor ligand-binding domain
1U3R Crystal Structure of Estrogen Receptor beta complexed with WAY-338 C A Nuclear receptor ligand-binding domain
1TFC CRYSTAL STRUCTURE OF THE LIGAND-BINDING DOMAIN OF THE ESTROGEN-RELATED RECEPTOR GAMMA IN COMPLEX WITH A STEROID RECEPTOR COACTIVATOR-1 PEPTIDE D B Nuclear receptor ligand-binding domain
1T7R Crystal structure of the androgen receptor ligand binding domain in complex with a FxxLF motif B A Nuclear receptor ligand-binding domain
1T76 Crystal structure of the androgen receptor ligand binding domain in complex with a WxxVW motif B A Nuclear receptor ligand-binding domain
1T79 Crystal structure of the androgen receptor ligand binding domain in complex with a FxxLW motif B A Nuclear receptor ligand-binding domain
1T7F Crystal structure of the androgen receptor ligand binding domain in complex with a LxxLL motif B A Nuclear receptor ligand-binding domain
1T7M Crystal structure of the androgen receptor ligand binding domain in complex with a FxxYF motif B A Nuclear receptor ligand-binding domain
1T74 Crystal structure of the androgen receptor ligand binding domain in complex with a WxxLF motif B A Nuclear receptor ligand-binding domain
1T73 Crystal structure of the androgen receptor ligand binding domain in complex with a FxxFF motif B A Nuclear receptor ligand-binding domain
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