 |
1A1R |
HCV NS3 PROTEASE DOMAIN:NS4A PEPTIDE COMPLEX |
C |
DAB |
Trypsin-like serine proteases |
|
 |
1AB9 |
CRYSTAL STRUCTURE OF BOVINE GAMMA-CHYMOTRYPSIN |
D |
CB |
|
|
 |
1AD8 |
COMPLEX OF THROMBIN WITH AND INHIBITOR CONTAINING A NOVEL P1 MOIETY |
L |
H |
|
|
 |
1B7X |
STRUCTURE OF HUMAN ALPHA-THROMBIN Y225I MUTANT BOUND TO D-PHE-PRO-ARG-CHLOROMETHYLKETONE |
A |
B |
|
|
 |
1BBR |
THE STRUCTURE OF RESIDUES 7-16 OF THE A ALPHA CHAIN OF HUMAN FIBRINOGEN BOUND TO BOVINE THROMBIN AT 2.3 ANGSTROMS RESOLUTION |
F |
HE |
|
|
 |
1BCU |
ALPHA-THROMBIN COMPLEXED WITH HIRUGEN AND PROFLAVIN |
L |
H |
|
|
 |
1BHX |
X-RAY STRUCTURE OF THE COMPLEX OF HUMAN ALPHA THROMBIN WITH THE INHIBITOR SDZ 229-357 |
E |
B |
|
|
 |
1CA0 |
BOVINE CHYMOTRYPSIN COMPLEXED TO APPI |
A |
CB |
|
|
 |
1DXP |
INHIBITION OF THE HEPATITIS C VIRUS NS3/4A PROTEASE. THE CRYSTAL STRUCTURES OF TWO PROTEASE-INHIBITOR COMPLEXES (APO STRUCTURE) |
C |
A |
Trypsin-like serine proteases |
|
 |
1DY8 |
INHIBITION OF THE HEPATITIS C VIRUS NS3/4A PROTEASE. THE CRYSTAL STRUCTURES OF TWO PROTEASE-INHIBITOR COMPLEXES (INHIBITOR II) |
C |
A |
Trypsin-like serine proteases |
|
 |
1DY9 |
INHIBITION OF THE HEPATITIS C VIRUS NS3/4A PROTEASE. THE CRYSTAL STRUCTURES OF TWO PROTEASE-INHIBITOR COMPLEXES (INHIBITOR I) |
C |
A |
Trypsin-like serine proteases |
|
 |
1GL1 |
STRUCTURE OF THE COMPLEX BETWEEN BOVINE ALPHA-CHYMOTRYPSIN AND PMP-C, AN INHIBITOR FROM THE INSECT LOCUSTA MIGRATORIA |
J |
B |
Trypsin-like serine proteases |
|
 |
1H8D |
X-RAY STRUCTURE OF THE HUMAN ALPHA-THROMBIN COMPLEX WITH A TRIPEPTIDE PHOSPHONATE INHIBITOR. |
L |
H |
|
|
 |
1H8I |
X-RAY CRYSTAL STRUCTURE OF HUMAN ALPHA-THROMBIN WITH A TRIPEPTIDE PHOSPHONATE INHIBITOR. |
L |
H |
|
|
 |
1HBT |
HUMAN ALPHA-THROMBIN COMPLEXED WITH A PEPTIDYL PYRIDINIUM METHYL KETONE CONTAINING BIVALENT INHIBITOR |
L |
H |
|
|
 |
1LHC |
HUMAN ALPHA-THROMBIN COMPLEXED WITH AC-(D)PHE-PRO-BOROARG-OH |
I |
H |
|
|
 |
1LHD |
HUMAN ALPHA-THROMBIN COMPLEXED WITH AC-(D)PHE-PRO-BOROLYS-OH |
I |
H |
|
|
 |
1LHE |
HUMAN ALPHA-THROMBIN COMPLEXED WITH AC-(D)PHE-PRO-BORO-N-BUTYL-AMIDINO-GLYCINE-OH |
I |
H |
|
|
 |
1LHF |
HUMAN ALPHA-THROMBIN COMPLEXED WITH AC-(D)PHE-PRO-BORO-HOMOLYS-OH |
I |
H |
|
|
 |
1LHG |
HUMAN ALPHA-THROMBIN COMPLEXED WITH AC-(D)PHE-PRO-BOROORNITHINE-OH |
I |
H |
|
|
 |
1MKW |
THE CO-CRYSTAL STRUCTURE OF UNLIGANDED BOVINE ALPHA-THROMBIN AND PRETHROMBIN-2: MOVEMENT OF THE YPPW SEGMENT AND ACTIVE SITE RESIDUES UPON LIGAND BINDING |
L |
H |
|
|
 |
1MKX |
THE CO-CRYSTAL STRUCTURE OF UNLIGANDED BOVINE ALPHA-THROMBIN AND PRETHROMBIN-2: MOVEMENT OF THE YPPW SEGMENT AND ACTIVE SITE RESIDUES UPON LIGAND BINDING |
L |
H |
|
|
 |
1O3P |
Elaborate Manifold of Short Hydrogen Bond Arrays Mediating Binding of Active Site-Directed Serine Protease Inhibitors |
A |
B |
|
|
 |
1R9N |
Crystal Structure of human dipeptidyl peptidase IV in complex with a decapeptide (tNPY) at 2.3 Ang. Resolution |
H |
D |
alpha/beta-Hydrolases |
|
 |
1RTF |
COMPLEX OF BENZAMIDINE WITH THE CATALYTIC DOMAIN OF HUMAN TWO CHAIN TISSUE PLASMINOGEN ACTIVATOR [(TC)-T-PA] |
A |
B |
|
|
 |
1SFQ |
Fast form of thrombin mutant R(77a)A bound to PPACK |
D |
E |
|
|
 |
1SHH |
Slow form of Thrombin Bound with PPACK |
A |
BE |
|
|
 |
1THP |
STRUCTURE OF HUMAN ALPHA-THROMBIN Y225P MUTANT BOUND TO D-PHE-PRO-ARG-CHLOROMETHYLKETONE |
A |
B |
|
|
 |
1TMT |
CHANGES IN INTERACTIONS IN COMPLEXES OF HIRUDIN DERIVATIVES AND HUMAN ALPHA-THROMBIN DUE TO DIFFERENT CRYSTAL FORMS |
J |
H |
|
|
 |
1TOM |
ALPHA-THROMBIN COMPLEXED WITH HIRUGEN |
L |
H |
|
|
 |
1UHB |
Crystal structure of porcine alpha trypsin bound with auto catalyticaly produced native peptide at 2.15 A resolution |
P |
BA |
Trypsin-like serine proteases |
|
 |
1UVT |
BOVINE THROMBIN--BM14.1248 COMPLEX |
L |
H |
|
|
 |
1VGC |
GAMMA-CHYMOTRYPSIN L-PARA-CHLORO-1-ACETAMIDO BORONIC ACID INHIBITOR COMPLEX |
A |
CB |
|
|
 |
1VZQ |
COMPLEX OF THROMBIN WITH DESIGNED INHIBITOR 7165 |
I |
H |
|
|
 |
1W3C |
CRYSTAL STRUCTURE OF THE HEPATITIS C VIRUS NS3 PROTEASE IN COMPLEX WITH A PEPTIDOMIMETIC INHIBITOR |
C |
A |
Trypsin-like serine proteases |
|
 |
1W7G |
ALPHA-THROMBIN COMPLEX WITH SULFATED HIRUDIN (RESIDUES 54-65) AND L-ARGININE TEMPLATE INHIBITOR CS107 |
L |
H |
|
|
 |
1WAY |
ACTIVE SITE THROMBIN INHIBITORS |
A |
B |
|
|
 |
1WBG |
ACTIVE SITE THROMBIN INHIBITORS |
A |
B |
|
|
 |
1YPH |
High resolution structure of bovine alpha-chymotrypsin |
A |
EC |
|
|
 |
2A0Q |
Structure of thrombin in 400 mM potassium chloride |
C |
D |
|
|
 |
2A2X |
Orally Active Thrombin Inhibitors in Complex with Thrombin Inh12 |
L |
H |
|
|
 |
2ANK |
orally active thrombin inhibitors in complex with thrombin and an exosite decapeptide |
L |
H |
|
|
 |
2BVR |
HUMAN THROMBIN COMPLEXED WITH FRAGMENT-BASED SMALL MOLECULES OCCUPYING THE S1 POCKET |
L |
H |
|
|
 |
2BVS |
HUMAN THROMBIN COMPLEXED WITH FRAGMENT-BASED SMALL MOLECULES OCCUPYING THE S1 POCKET |
L |
H |
|
|
 |
2C8W |
THROMBIN INHIBITORS |
A |
B |
|
|
 |
2C8Y |
THROMBIN INHIBITORS |
A |
B |
|
|
 |
2C8Z |
THROMBIN INHIBITORS |
A |
B |
|
|
 |
2C90 |
THROMBIN INHIBITORS |
A |
B |
|
|
 |
2C93 |
THROMBIN INHIBITORS |
A |
B |
|
|
 |
2CF8 |
COMPLEX OF RECOMBINANT HUMAN THROMBIN WITH A INHIBITOR |
I |
H |
|
|