 |
1GWQ |
HUMAN OESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH RALOXIFENE CORE AND TIF2 NRBOX2 PEPTIDE |
C |
A |
Nuclear receptor ligand-binding domain |
|
 |
1GWR |
HUMAN OESTROGEN RECEPTOR ALPHA LIGAND-BINDING DOMAIN IN COMPLEX WITH 17BETA-OESTRADIOL AND TIF2 NRBOX3 PEPTIDE |
C |
A |
Nuclear receptor ligand-binding domain |
|
 |
1YCQ |
XENOPUS LAEVIS MDM2 BOUND TO THE TRANSACTIVATION DOMAIN OF HUMAN P53 |
B |
A |
SWIB/MDM2 domain |
|
 |
2BJ4 |
ESTROGEN RECEPTOR ALPHA LBD IN COMPLEX WITH A PHAGE-DISPLAY DERIVED PEPTIDE ANTAGONIST |
C |
A |
|
|
 |
2J7X |
STRUCTURE OF ESTRADIOL-BOUND ESTROGEN RECEPTOR BETA LBD IN COMPLEX WITH LXXLL MOTIF FROM NCOA5 |
B |
A |
Nuclear receptor ligand-binding domain |
|
 |
2J7Y |
STRUCTURE OF 17-EPIESTRIOL-BOUND ESTROGEN RECEPTOR BETA LBD IN COMPLEX WITH LXXLL MOTIF FROM NCOA5 |
B |
A |
Nuclear receptor ligand-binding domain |
|
 |
2JF9 |
ESTROGEN RECEPTOR ALPHA LBD IN COMPLEX WITH A TAMOXIFEN-SPECIFIC PEPTIDE ANTAGONIST |
P |
AC |
|
|
 |
2QPY |
AR LBD with small molecule |
B |
A |
Nuclear receptor ligand-binding domain |
|
 |
2QR9 |
Crystal Structure of the Estrogen Receptor Alpha Ligand Binding Domain Complexed with an Oxabicyclic Derivative Compound |
C |
A |
|
|
 |
2QSE |
Crystal Structure of the Estrogen Receptor Alpha Ligand Binding Domain complexed with Burned Meat Compound 4-OH-PhIP |
C |
A |
|
|
 |
2QXM |
Crystal Structure of the Estrogen Receptor Alpha Ligand Binding Domain Complexed to Burned Meat Compound PhIP |
C |
A |
|
|
 |
2QXV |
Structural basis of EZH2 recognition by EED |
B |
A |
|
|
 |
2QZO |
Crystal Structure of the Estrogen Receptor Alpha Ligand Binding Domain Complexed with WAY-169916 |
C |
A |
|
|
 |
2W9R |
STRUCTURAL BASIS OF N-END RULE SUBSTRATE RECOGNITION IN ESCHERICHIA COLI BY THE CLPAP ADAPTOR PROTEIN CLPS |
B |
A |
|
|
 |
2Z5S |
Molecular basis for the inhibition of p53 by Mdmx |
R |
O |
|
|
 |
2Z5T |
Molecular basis for the inhibition of p53 by Mdmx |
P |
MO |
|
|
 |
2ZFX |
Crystal structure of the rat vitamin D receptor ligand binding domain complexed with YR301 and a synthetic peptide containing the NR2 box of DRIP 205 |
C |
A |
|
|
 |
2ZL9 |
2-Substituted-16-ene-22-thia-1alpha,25-dihydroxy-26,27-dimethyl-19-norvitamin D3 analogs: Synthesis, biological evaluation and crystal structure |
C |
A |
Nuclear receptor ligand-binding domain |
|
 |
2ZLA |
2-Substituted-16-ene-22-thia-1alpha,25-dihydroxy-26,27-dimethyl-19-norvitamin D3 analogs: Synthesis, biological evaluation and crystal structure |
C |
A |
Nuclear receptor ligand-binding domain |
|
 |
2ZLC |
2-Substituted-16-ene-22-thia-1alpha,25-dihydroxy-26,27-dimethyl-19-norvitamin D3 analogs: Synthesis, biological evaluation and crystal structure |
C |
A |
Nuclear receptor ligand-binding domain |
|
 |
2ZMH |
Crystal Structure of Rat Vitamin D Receptor Bound to Adamantyl Vitamin D Analogs: Structural Basis for Vitamin D Receptor Antagonism and/or Partial Agonism |
C |
A |
Nuclear receptor ligand-binding domain |
|
 |
2ZMI |
Crystal Structure of Rat Vitamin D Receptor Bound to Adamantyl Vitamin D Analogs: Structural Basis for Vitamin D Receptor Antagonism and/or Partial Agonism |
C |
A |
Nuclear receptor ligand-binding domain |
|
 |
2ZMJ |
Crystal Structure of Rat Vitamin D Receptor Bound to Adamantyl Vitamin D Analogs: Structural Basis for Vitamin D Receptor Antagonism and/or Partial Agonism |
C |
A |
Nuclear receptor ligand-binding domain |
|
 |
2ZVV |
Crystal structure of Proliferating cellular nuclear antigen 1 and Short peptide from human P21 |
X |
YAB |
|
|
 |
2ZXN |
A New Class of Vitamin D Receptor Ligands that Induce Structural Rearrangement of the Ligand-binding Pocket |
C |
A |
|
|
 |
3BEJ |
Structure of human FXR in complex with MFA-1 and co-activator peptide |
E |
A |
Nuclear receptor ligand-binding domain |
|
 |
3BQD |
Doubling the Size of the Glucocorticoid Receptor Ligand Binding Pocket by Deacylcortivazol |
B |
A |
Nuclear receptor ligand-binding domain |
|
 |
3BQO |
Crystal Structure of TRF1 TRFH domain and TIN2 peptide complex |
B |
A |
Telomeric repeat binding factor (TRF) dimerisation domain |
|
 |
3BU8 |
Crystal Structure of TRF2 TRFH domain and TIN2 peptide complex |
D |
B |
Telomeric repeat binding factor (TRF) dimerisation domain |
|
 |
3BUA |
Crystal Structure of TRF2 TRFH domain and APOLLO peptide complex |
F |
B |
Telomeric repeat binding factor (TRF) dimerisation domain |
|
 |
3C2G |
Crystal complex of SYS-1/POP-1 at 2.5A resolution |
C |
A |
|
|
 |
3CS8 |
Structural and Biochemical Basis for the Binding Selectivity of PPARg to PGC-1a |
B |
A |
Nuclear receptor ligand-binding domain |
|
 |
3CWD |
Molecular recognition of nitro-fatty acids by PPAR gamma |
C |
A |
Nuclear receptor ligand-binding domain |
|
 |
3D24 |
Crystal structure of ligand-binding domain of estrogen-related receptor alpha (ERRalpha) in complex with the peroxisome proliferators-activated receptor coactivator-1alpha box3 peptide (PGC-1alpha) |
B |
A |
Nuclear receptor ligand-binding domain |
|
 |
3DAB |
Structure of the human Mdmx protein bound to the p53 tumor suppressor transactivation domain |
D |
C |
|
|
 |
3DAC |
Structure of the human Mdmx protein bound to the p53 tumor suppressor transactivation domain |
P |
M |
|
|
 |
3DCT |
FXR with SRC1 and GW4064 |
B |
A |
Nuclear receptor ligand-binding domain |
|
 |
3E7C |
Glucocorticoid Receptor LBD bound to GSK866 |
D |
B |
|
|
 |
3E94 |
Crystal structure of RXRalpha ligand binding domain in complex with tributyltin and a coactivator fragment |
B |
A |
|
|
 |
3ECH |
The MarR-family repressor MexR in complex with its antirepressor ArmR |
C |
BA |
|
|
 |
3ET1 |
Structure of PPARalpha with 3-[5-Methoxy-1-(4-methoxy-benzenesulfonyl)-1H-indol-3-yl]-propionic acid |
P |
A |
|
|
 |
3ET3 |
Structure of PPARgamma with 3-[5-Methoxy-1-(4-methoxy-benzenesulfonyl)-1H-indol-3-yl]-propionic acid |
P |
A |
|
|
 |
3F7D |
SF-1 LBD bound by phosphatidylcholine |
B |
A |
|
|
 |
3F9W |
Structural Insights into Lysine Multiple Methylation by SET Domain Methyltransferases, SET8-Y334F / H4-Lys20 / AdoHcy |
F |
AB |
|
|
 |
3F9Z |
Structural Insights into Lysine Multiple Methylation by SET Domain Methyltransferases, SET8-Y245F / H4-Lys20 / AdoHcy |
G |
A |
|
|
 |
3FUG |
Crystal Structure of the Retinoid X Receptor Ligand Binding Domain Bound to the Synthetic Agonist 3-[4-Hydroxy-3-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaphthalen-2-yl)-phenyl]acrylic Acid |
B |
A |
|
|
 |
3FUR |
Crystal Structure of PPARg in complex with INT131 |
H |
A |
|
|
 |
3FXV |
Identification of an N-oxide pyridine GW4064 analogue as a potent FXR agonist |
B |
A |
|
|
 |
3G8I |
Aleglitazar, a new, potent, and balanced PPAR alpha/gamma agonist for the treatment of type II diabetes |
Z |
A |
|
|
 |
3G9E |
Aleglitaar. a new. potent, and balanced dual ppara/g agonist for the treatment of type II diabetes |
B |
A |
|
|