 |
1APM |
2.0 ANGSTROM REFINED CRYSTAL STRUCTURE OF THE CATALYTIC SUBUNIT OF CAMP-DEPENDENT PROTEIN KINASE COMPLEXED WITH A PEPTIDE INHIBITOR AND DETERGENT |
I |
E |
Protein kinase-like (PK-like) |
|
 |
1CDK |
CAMP-DEPENDENT PROTEIN KINASE CATALYTIC SUBUNIT (E.C.2.7.1.37) (PROTEIN KINASE A) COMPLEXED WITH PROTEIN KINASE INHIBITOR PEPTIDE FRAGMENT 5-24 (PKI(5-24) ISOELECTRIC VARIANT CA) AND MN2+ ADENYLYL IMIDODIPHOSPHATE (MNAMP-PNP) AT PH 5.6 AND 7C AND 4C |
I |
A |
Protein kinase-like (PK-like) |
|
 |
1FMO |
CRYSTAL STRUCTURE OF A POLYHISTIDINE-TAGGED RECOMBINANT CATALYTIC SUBUNIT OF CAMP-DEPENDENT PROTEIN KINASE COMPLEXED WITH THE PEPTIDE INHIBITOR PKI(5-24) AND ADENOSINE |
I |
E |
Protein kinase-like (PK-like) |
|
 |
1IR3 |
PHOSPHORYLATED INSULIN RECEPTOR TYROSINE KINASE IN COMPLEX WITH PEPTIDE SUBSTRATE AND ATP ANALOG |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1K3A |
Structure of the Insulin-like Growth Factor 1 Receptor Kinase |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1LEW |
CRYSTAL STRUCTURE OF MAP KINASE P38 COMPLEXED TO THE DOCKING SITE ON ITS NUCLEAR SUBSTRATE MEF2A |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1LEZ |
CRYSTAL STRUCTURE OF MAP KINASE P38 COMPLEXED TO THE DOCKING SITE ON ITS ACTIVATOR MKK3B |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1NVQ |
The Complex Structure Of Checkpoint Kinase Chk1/UCN-01 |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1NVR |
The Complex Structure Of Checkpoint Kinase Chk1/Staurosporine |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1NVS |
The Complex Structure Of Checkpoint Kinase Chk1/SB218078 |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1O6K |
STRUCTURE OF ACTIVATED FORM OF PKB KINASE DOMAIN S474D WITH GSK3 PEPTIDE AND AMP-PNP |
C |
A |
Protein kinase-like (PK-like) |
|
 |
1O6L |
CRYSTAL STRUCTURE OF AN ACTIVATED AKT/PROTEIN KINASE B (PKB-PIF CHIMERA) TERNARY COMPLEX WITH AMP-PNP AND GSK3 PEPTIDE |
C |
A |
Protein kinase-like (PK-like) |
|
 |
1O9U |
GLYCOGEN SYNTHASE KINASE 3 BETA COMPLEXED WITH AXIN PEPTIDE |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1Q61 |
PKA triple mutant model of PKB |
I |
A |
Protein kinase-like (PK-like) |
|
 |
1Q62 |
PKA double mutant model of PKB |
I |
A |
Protein kinase-like (PK-like) |
|
 |
1Q8T |
The Catalytic Subunit of cAMP-dependent Protein Kinase (PKA) in Complex with Rho-kinase Inhibitor Y-27632 |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1Q8U |
The Catalytic Subunit of cAMP-dependent Protein Kinase in Complex with Rho-kinase Inhibitor H-1152P |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1Q8W |
The Catalytic Subunit of cAMP-dependent Protein Kinase in Complex with Rho-kinase Inhibitor Fasudil (HA-1077) |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1QMZ |
PHOSPHORYLATED CDK2-CYCLYIN A-SUBSTRATE PEPTIDE COMPLEX |
E |
C |
Protein kinase-like (PK-like) |
|
 |
1SMH |
Protein kinase A variant complex with completely ordered N-terminal helix |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1STC |
CAMP-DEPENDENT PROTEIN KINASE, ALPHA-CATALYTIC SUBUNIT IN COMPLEX WITH STAUROSPORINE |
I |
E |
Protein kinase-like (PK-like) |
|
 |
1SVE |
Crystal Structure of Protein Kinase A in Complex with Azepane Derivative 1 |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1SVG |
Crystal Structure of Protein Kinase A in Complex with Azepane Derivative 4 |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1SVH |
Crystal Structure of Protein Kinase A in Complex with Azepane Derivative 8 |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1UKH |
Structural basis for the selective inhibition of JNK1 by the scaffolding protein JIP1 and SP600125 |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1XH4 |
Crystal Structures of Protein Kinase B Selective Inhibitors in Complex with Protein Kinase A and Mutants |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1XH5 |
Crystal Structures of Protein Kinase B Selective Inhibitors in Complex with Protein Kinase A and Mutants |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1XH6 |
Crystal Structures of Protein Kinase B Selective Inhibitors in Complex with Protein Kinase A and Mutants |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1XH7 |
Crystal Structures of Protein Kinase B Selective Inhibitors in Complex with Protein Kinase A and Mutants |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1XH8 |
Crystal Structures of Protein Kinase B Selective Inhibitors in Complex with Protein Kinase A and Mutants |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1XH9 |
Crystal Structures of Protein Kinase B Selective Inhibitors in Complex with Protein Kinase A and Mutants |
B |
A |
|
|
 |
1XHA |
Crystal Structures of Protein Kinase B Selective Inhibitors in Complex with Protein Kinase A and Mutants |
B |
A |
Protein kinase-like (PK-like) |
|
 |
1YDR |
STRUCTURE OF CAMP-DEPENDENT PROTEIN KINASE, ALPHA-CATALYTIC SUBUNIT IN COMPLEX WITH H7 PROTEIN KINASE INHIBITOR 1-(5-ISOQUINOLINESULFONYL)-2-METHYLPIPERAZINE |
I |
E |
Protein kinase-like (PK-like) |
|
 |
1YDS |
STRUCTURE OF CAMP-DEPENDENT PROTEIN KINASE, ALPHA-CATALYTIC SUBUNIT IN COMPLEX WITH H8 PROTEIN KINASE INHIBITOR [N-(2-METHYLAMINO)ETHYL]-5-ISOQUINOLINESULFONAMIDE |
I |
E |
Protein kinase-like (PK-like) |
|
 |
1YDT |
STRUCTURE OF CAMP-DEPENDENT PROTEIN KINASE, ALPHA-CATALYTIC SUBUNIT IN COMPLEX WITH H89 PROTEIN KINASE INHIBITOR N-[2-(4-BROMOCINNAMYLAMINO)ETHYL]-5-ISOQUINOLINE |
I |
E |
Protein kinase-like (PK-like) |
|
 |
1ZYS |
Co-crystal structure of Checkpoint Kinase Chk1 with a pyrrolo-pyridine inhibitor |
B |
A |
|
|
 |
2BFY |
COMPLEX OF AURORA-B WITH INCENP AND HESPERIDIN. |
D |
A |
|
|
 |
2BZK |
CRYSTAL STRUCTURE OF THE HUMAN PIM1 IN COMPLEX WITH AMPPNP AND PIMTIDE |
A |
B |
|
|
 |
2C1A |
STRUCTURE OF CAMP-DEPENDENT PROTEIN KINASE COMPLEXED WITH ISOQUINOLINE-5-SULFONIC ACID (2-(2-(4-CHLOROBENZYLOXY) ETHYLAMINO)ETHYL)AMIDE |
I |
A |
Protein kinase-like (PK-like) |
|
 |
2C1B |
STRUCTURE OF CAMP-DEPENDENT PROTEIN KINASE COMPLEXED WITH (4R,2S)-5\'-(4-(4-CHLOROBENZYLOXY)PYRROLIDIN-2-YLMETHANESULFONYL)ISOQUINOLINE |
I |
A |
Protein kinase-like (PK-like) |
|
 |
2C3I |
CRYSTAL STRUCTURE OF HUMAN PIM1 IN COMPLEX WITH IMIDAZOPYRIDAZIN I |
A |
B |
|
|
 |
2ERZ |
Crystal Structure of c-AMP Dependent Kinase (PKA) bound to hydroxyfasudil |
I |
E |
Protein kinase-like (PK-like) |
|
 |
2F7E |
PKA complexed with (S)-2-(1H-Indol-3-yl)-1-(5-isoquinolin-6-yl-pyridin-3-yloxymethyl-etylamine |
I |
E |
Protein kinase-like (PK-like) |
|
 |
2F7X |
Protein Kinase A bound to (S)-2-(1H-Indol-3-yl)-1-[5-((E)-2-pyridin-4-yl-vinyl)-pyridin-3-yloxymethyl]-ethylamine |
I |
E |
Protein kinase-like (PK-like) |
|
 |
2FYS |
Crystal structure of Erk2 complex with KIM peptide derived from MKP3 |
D |
BA |
Protein kinase-like (PK-like) |
|
 |
2GFC |
cAMP-dependent protein kinase PKA catalytic subunit with PKI-5-24 |
I |
A |
Protein kinase-like (PK-like) |
|
 |
2GNF |
Protein kinase A fivefold mutant model of Rho-kinase with Y-27632 |
I |
A |
|
|
 |
2GNG |
Protein kinase A fivefold mutant model of Rho-kinase |
I |
A |
|
|
 |
2GNH |
PKA five fold mutant model of Rho-kinase with H1152P |
I |
A |
|
|
 |
2GNI |
PKA fivefold mutant model of Rho-kinase with inhibitor Fasudil (HA1077) |
I |
A |
|
|